DPI-3290

DPI-3290

DPI-3290
Systematic (IUPAC) name
(+)-3-((αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl)-N-(3-fluorophenyl)-N-methylbenzamide
Identifiers
CAS Registry Number  N
PubChem CID:
Chemical data
Formula C30H34FN3O2
Molecular mass 487.607 g/mol
 N   

DPI-3290 was discovered by Delta Pharmaceutical [1] and is a drug that is used in scientific research. It is a potent analgesic drug,[2] which produces little respiratory depression.[3]

DPI-3290 acts as an agonist at both μ- and δ-opioid receptor, with an IC50 of 6.2nM at μ and 1.0nM at δ.[4]

References

  1. ^ US Patent 5552404 - Opioid compounds and methods for using same
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